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Supplements/Compound

Alpha-Lipoic Acid

aka ALA · R-ALA

Mitochondrial antioxidant studied for diabetic neuropathy and insulin sensitivity.

Overview

Mitochondrial antioxidant studied for diabetic neuropathy and insulin sensitivity.

Natural sources
  • Trace in red meat, organ meats
Common forms
  • Racemic ALA
  • R-ALA (active enantiomer)

Forms & variants of Alpha-Lipoic Acid

Different chemical forms of Alpha-Lipoic Acid behave differently. Browse each form's mechanism, bioavailability, and best-use context.

Mechanism of action

Cofactor for pyruvate and α-KG dehydrogenase; regenerates other antioxidants; activates AMPK.

Pathways
  • · AMPK activation
  • · Antioxidant recycling

Effects on the body

Decreases
Fasting glucose
Decreases
Diabetic neuropathy symptoms

Organ system effects

Brain & CNS

Reduces diabetic neuropathy pain.

Evidence-based benefits

Reduces diabetic neuropathy symptoms (600 mg/d)

Strong evidence

Potential side effects

Common
  • · Nausea
Rare
  • · Skin rash
Serious
  • · Insulin autoimmune syndrome (rare)

Drug interactions

Insulin / sulfonylureas
Hypoglycemia risk.
moderate
Thyroid hormone
May reduce conversion.
minor

Safety & non-supplemental interactions

Educational summary — always confirm with your clinician or pharmacist before starting, stopping, or combining with prescription therapy.

Avoid with these conditions
  • ·Thiamine deficiency (e.g. alcohol-use disorder)
  • ·Thyroid disorders
Avoid / monitor with these medications
  • ·Insulin and antidiabetic drugs (hypoglycemia)
  • ·Thyroid hormone (reduced absorption)
  • ·Chemotherapy

Supplement interactions

Pairs well with

None listed.

Avoid combining with

No specific avoidances listed.

Dosing & bioavailability

Typical dose
300–600 mg R-ALA or 600–1800 mg racemic

Where to buy

Affiliate-style search links to reputable retailers. We don't endorse specific brands — verify third-party testing (USP, NSF, Informed Sport) before purchase.

Scientific evidence (8)

RCTDiabetes Care · 2006

ALA for diabetic peripheral neuropathy (SYDNEY 2)

Ziegler D, et al.

5-week RCT of oral ALA in diabetic neuropathy.

Key findings

Significant symptom and neuropathic-impairment improvement.

Open study
Systematic reviewPubMed (NLM) · 1970

PubMed: Alpha-Lipoic Acid — Reduces diabetic neuropathy symptoms

Live PubMed search

Live results for "Alpha-Lipoic Acid Reduces diabetic neuropathy symptoms" across the PubMed/MEDLINE peer-reviewed index.

Key findings

Opens current human and preclinical literature matching Alpha-Lipoic Acid and "Reduces diabetic neuropathy symptoms". Filter by RCT, meta-analysis, or year on the results page.

Open study
Systematic reviewPubMed (NLM) · 1970

PubMed: Alpha-Lipoic Acid — randomized controlled trial

Live PubMed search

Live results for "Alpha-Lipoic Acid randomized controlled trial" across the PubMed/MEDLINE peer-reviewed index.

Key findings

Opens current human and preclinical literature matching Alpha-Lipoic Acid and "randomized controlled trial". Filter by RCT, meta-analysis, or year on the results page.

Open study
Systematic reviewPubMed (NLM) · 1970

PubMed: Alpha-Lipoic Acid — meta-analysis

Live PubMed search

Live results for "Alpha-Lipoic Acid meta-analysis" across the PubMed/MEDLINE peer-reviewed index.

Key findings

Opens current human and preclinical literature matching Alpha-Lipoic Acid and "meta-analysis". Filter by RCT, meta-analysis, or year on the results page.

Open study
Systematic reviewPubMed (NLM) · 1970

PubMed: Alpha-Lipoic Acid — pharmacokinetics

Live PubMed search

Live results for "Alpha-Lipoic Acid pharmacokinetics" across the PubMed/MEDLINE peer-reviewed index.

Key findings

Opens current human and preclinical literature matching Alpha-Lipoic Acid and "pharmacokinetics". Filter by RCT, meta-analysis, or year on the results page.

Open study
Systematic reviewPubMed (NLM) · 1970

PubMed: Alpha-Lipoic Acid — safety adverse events

Live PubMed search

Live results for "Alpha-Lipoic Acid safety adverse events" across the PubMed/MEDLINE peer-reviewed index.

Key findings

Opens current human and preclinical literature matching Alpha-Lipoic Acid and "safety adverse events". Filter by RCT, meta-analysis, or year on the results page.

Open study
Systematic reviewPubMed (NLM) · 1970

PubMed: Alpha-Lipoic Acid — dose response

Live PubMed search

Live results for "Alpha-Lipoic Acid dose response" across the PubMed/MEDLINE peer-reviewed index.

Key findings

Opens current human and preclinical literature matching Alpha-Lipoic Acid and "dose response". Filter by RCT, meta-analysis, or year on the results page.

Open study
Systematic reviewGoogle Scholar · 1970

Google Scholar: Alpha-Lipoic Acid — clinical evidence

Live Scholar search

Cross-database citation index for Alpha-Lipoic Acid as it relates to "clinical evidence".

Key findings

Includes preprints, theses, and journal articles. Useful for tracking citation counts and follow-on work.

Open study
Educational use only. This profile is not medical advice. Consult a qualified healthcare professional before starting any supplement, especially if you take prescription medication or have a chronic condition.